发明名称 Crystalline diastereomeric L-alpha-methyldopa POE ester and process for its preparation
摘要 Disclosed is a crystalline form of diastereomeric L- alpha -methyldopa POE ester, also referred to as (R),(S)- alpha -pivaloyloxyethyl-(S)-3-(3,4-dihydroxyphenyl)-2-methylalaninate and a process for its isolation. Also disclosed is an improved process for the formation of diastereomeric L- alpha -methyldopa POE ester.
申请公布号 US4440942(A) 申请公布日期 1984.04.03
申请号 US19820353697 申请日期 1982.03.01
申请人 MERCK & CO., INC. 发明人 BUDAVARI, JOHN
分类号 C07C227/34;C07C67/00;C07C227/00;C07C227/18;C07C227/42;C07C229/36;(IPC1-7):C07C101/08 主分类号 C07C227/34
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