N-formyl and n-hydroxymethyl-3-phenoxy-1-azetidinecarboxamides and their preparation and use.

摘要

N-Formyl and N-hydroxymethy)-3-phenoxy-1-azetidinecarboxamides having the formula:
<Chemistry id="chema01" num="0001"><Image id="ia01" he="17" wi="64" file="IMGA0001.TIF" imgContent="chem" imgFormat="TIFF" inline="no" /></Chemistry>wherein R is selected from formyl and hydroxymethyl and R' is selected from hydrogen, fluoro, loweralkyl, lower-alkoxy, trifluoromethyl, acetyl, N-formylcarboxamido or N-hydroxymethylcarboxamido having anticonvulsant activity are disclosed.