发明名称 AMIDINER
摘要 Mitomycin A, mitomycin C, and porfiromycin react with amide acetals and other amide derivatives to produce amidine derivatives having antitumor activity against experimental animal tumors. The amidines derived from mitomycin C are useful intermediates in reactions with primary amines to produce both known and novel 7-amino-9a-methoxymitosanes having antitumor activity against experimental animal tumors.
申请公布号 FI831972(L) 申请公布日期 1983.12.05
申请号 FI19830001972 申请日期 1983.06.01
申请人 BRISTOL-MYERS COMPANY 发明人 VYAS, DOLATRAI MOHANLAL;KANEKO, TAKUSHI;DOYLE, TERRENCE WILLIAM
分类号 C07D487/14 主分类号 C07D487/14
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