| 发明名称 |
A PROCESS FOR PREPARING [1S- ]1-ALPHA, 2-ALPHA, 3-BETA (1S, 2R) 5- BETA] ]-3- [7- [2- (3, 4-DIF LUOROPHENYL) -CYCLOPROPYLAMINO]- 5- (PROPYLTHIO) -3H-1, 2, 3-TRIAZOLO [4, 5-D]PYRIMIDIN-3-YL]-5- (2- HYDROXYETHOXY) CYCLOPENTANE-1, 2-DIOL AND TO ITS INTERMEDIATES [1S-[123(1S2R)5]]-3-[7-[2-(34-)-]- 5-()-3H-123-[45-D]-3-]-5-(2-)-12- |
| 摘要 |
The present invention is directed to a process for preparing [1S-[1alpha,2alpha,3beta(1S*,2R*),5beta]]-3-[7-[2-(3,4-difluorophenyl)-cyclopropylamino]-5-(propylthio)-3H-1,2,3-triazolo[4,5-d]pyrimidin-3-yl]-5-(2-hydroxyethoxy)cyclopentane-1,2-diol and to intermediates useful in the process. |
| 申请公布号 |
HK1159103(A1) |
申请公布日期 |
2016.09.15 |
| 申请号 |
HK20110113635 |
申请日期 |
2011.12.16 |
| 申请人 |
ASTRAZENECA AB |
发明人 |
AUFDENBLATTEN, Rhony;BOHLIN, Martin, Hans;HELLSTRM, Helena;JOHANSSON, Peter, W;LARSSON, Ulf, G;RECKNAGEL, Mikaela;WEISS, Ursula, heiress of WEISS Andreas |
| 分类号 |
C07D |
主分类号 |
C07D |
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