发明名称 PROCESS FOR THE PREPARATION OF 5'-DEOXY-5-FLUORO URIDINE AND INTERMEDIATES IN THIS PROCESS
摘要 A process for the manufacture of 5'-deoxy-5-fluorouridine which is a potent antitumor agent. The process comprises cleaving the acyl groups from a 1-(5-deoxy-2,3-di-O-acyl- beta -D-ribofuranosyl)-5-fluorouracil, a novel intermediate in the process.
申请公布号 EP0021231(B1) 申请公布日期 1983.10.05
申请号 EP19800103219 申请日期 1980.06.10
申请人 F. HOFFMANN-LA ROCHE & CO. AKTIENGESELLSCHAFT 发明人 D'SOUSA, RICHARD;KISS, JOSEPH, PROF. DR.
分类号 C07H19/067;C07H15/04;C07H19/06 主分类号 C07H19/067
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