发明名称 PROCEDIMIENTO PARA LA PREPARACION DE DERIVADOS DEL ACIDO CIS, ENDO-2-AZABICICLO (3.3.0)-OCTAN-3-CARBOXILICO.
摘要 <p>Compounds of the formula I <IMAGE> (I) in which the carboxyl group on carbon atom 3 is orientated in the endo-position relative to the bicyclic ring system of cis-configuration, and in which R1 denotes hydrogen, allyl, vinyl or a side-chain of a naturally occurring alpha -aminoacid, which may be protected, R2 denotes hydrogen, alkyl, alkenyl or aralkyl, Y denotes hydrogen or hydroxyl and Z denotes hydrogen, or Y and Z together denote oxygen, and X denotes alkyl, alkenyl or cycloalkyl, or aryl which is optionally mono-, di- or tri-substituted by alkyl, alkoxy, hydroxyl, halogen, nitro, amino, alkylamino, dialkylamino or methylenedioxy, or denotes indol-3-yl, a process for their preparation, agents containing these compounds and their use.</p>
申请公布号 ES517066(D0) 申请公布日期 1983.08.01
申请号 ES19660005170 申请日期 1982.11.03
申请人 HOECHST AKTIENGESELLSCHAFT 发明人
分类号 C07C227/08;A61K31/40;A61K31/403;A61K38/00;A61P9/12;C07C227/10;C07C227/16;C07C229/36;C07C237/06;C07D209/52;C07D451/04;C07K5/02;C07K5/06;(IPC1-7):07D209/02;61K31/40;07D209/52;61K31/435 主分类号 C07C227/08
代理机构 代理人
主权项
地址