发明名称 |
Inhibition of GABA uptake by N-substituted azaheterocyclic carboxylic acids and their esters |
摘要 |
N-Substituted azaheterocyclic carboxylic acids and their esters, useful as inhibitors of GABA uptake, are prepared by reacting an appropriate N-alkylating derivative with an ester of an N-unsubstituted azaheterocyclic carboxylic acid followed by hydrolysis of the ester.
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申请公布号 |
US4383999(A) |
申请公布日期 |
1983.05.17 |
申请号 |
US19820372504 |
申请日期 |
1982.04.28 |
申请人 |
SMITHKLINE BECKMAN CORPORATION |
发明人 |
BONDINELL, WILLIAM E.;LAFFERTY, JOHN J.;ZIRKLE, CHARLES L. |
分类号 |
C07C17/16;C07C17/26;C07C43/178;C07C45/00;C07D211/34;C07D211/60;C07D211/78;(IPC1-7):A61K31/45;A61K31/44 |
主分类号 |
C07C17/16 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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