发明名称 |
FOERFARANDE FOER FRAMSTAELLNING AV ULCUSHAEMMANDE N-SUBSTITUERADE 5,11-DIHYDRO-6H-PYRIDO(2,3-B)(1,4)BENSODIAZEPIN-6-ONER |
摘要 |
<p>Compounds of the formula <IMAGE> wherein R1 is alkyl of 3 to 12 carbon atoms; unsaturated aliphatic hydrocarbyl of 3 to 20 carbon atoms comprising 1 to 3 double bonds and/or one triple bond; phenyl(alkyl of 2 to 4 carbon atoms); methylenedioxybenzyl; chlorobenzyl; indan-5-ylmethyl; indan-3-ylmethyl; phenyl(alkenyl of 2 to 4 carbon atoms); cycloalkyl of 5 to 7 carbon atoms; (cycloalkyl of 3 to 10 carbon atoms)methyl; (methylcycloalkyl of 4 to 11 carbon atoms)methyl; morpholino(alkyl of 2 to 3 carbon atoms); pyrrolidino(alkyl of 2 to 3 carbon atoms); piperidino (alkyl of 2 to 3 carbon atoms); 4-methylpiperazino(alkyl of 2 to 3 carbon atoms); or, when R3 and/or R4 are methyl or ethyl, also methyl or ethyl; R2 is hydrogen, methyl or ethyl; and R3 and R4 are each hydrogen, methyl or ethyl; and non-toxic, pharmacologically acceptable acid addition salts thereof. The compounds as well as the salts are useful as anti-ulcerogenics and secretion inhibitors.</p> |
申请公布号 |
FI63232(C) |
申请公布日期 |
1983.05.10 |
申请号 |
FI19780001474 |
申请日期 |
1978.05.10 |
申请人 |
DR KARL THOMAE GMBH |
发明人 |
SCHMIDT GUENTHER;LEITOLD MATYAS |
分类号 |
A61K31/00;A61K31/5513;A61P1/04;A61P25/02;C07D471/04;(IPC1-7):C07D471/04 |
主分类号 |
A61K31/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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