发明名称 Processes for the preparation of cyanoheterocycles
摘要 Processes for the preparation of cyanoheterocycles of the general formula I <IMAGE> in which W, X, Y and Z denote a nitrogen atom or the radicals CH or CR1 where R1 denotes a hydrogen atom, a straight-chain or branched alkyl radical having 1-10 C atoms, which may be substituted, an aralkyl having 7-10 C atoms, aryl, heteroaryl, methoxycarbonyl, ethoxycarbonyl, phenoxycarbonyl, carboxyl, a hydroxyl radical, an amino radical, a mono- or dialkylamino radical, a mono- or diarylamino radical, alkylsulphonyl, arylsulphonyl, trifluoromethyl, a halogen substituent or a cycloalkyl, or W-X, X-Y and Y-Z form part of an aliphatic, aromatic or heterocyclic ring, which may contain one or more nitrogen, oxygen or sulphur atoms and be substituted by R1 where R1 has the meaning given, are characterised in that an N-oxide of the general formula II <IMAGE> in which W, X, Y, Z and R1 have the meanings given, is reacted with trimethylsilyl cyanide.
申请公布号 DE3141640(A1) 申请公布日期 1983.05.05
申请号 DE19813141640 申请日期 1981.10.16
申请人 SCHERING AG 发明人 VORBRUEGGEN,HELMUT,PROF.
分类号 C07D213/00;C07D213/84;C07D213/85;C07D215/48;C07D217/26;C07D521/00;(IPC1-7):C07D213/84;C07D239/28;C07D237/24;C07D241/24;C07D219/04;C07D471/04;C07D473/00 主分类号 C07D213/00
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