发明名称 PROCESS OF PREPARATION OF THIENO AND FURO-(2,3-C)PYRROLES
摘要 <p>Derivatives represented by the formula <IMAGE> in which X1 and X2 denote an oxygen or sulphur atom; R1 denotes a linear or branched alkyl radical containing from 1 to 8 carbon atoms, an alkynyl radical, an alkoxyalkyl radical containing from 3 to 8 carbon atoms or an aromatic residue; R2 denotes a hydrogen atom or a linear or branched alkyl radical; m = 2 or 3, when m = 2, X1 and X2 denote a sulphur atom. U denotes a 3,4-diaminocyclobuten-1,2-dione or aminosulphonylformamidine residue; U may also denote the nitrogenous structures <IMAGE> in which V denotes a nitrogen atom or a CH fragment; W denotes NO2 or CN; R3 denotes a hydrogen atom, a linear or branched alkyl radical containing 1 to 8 carbon atoms, or an alkynyl radical; R4 denotes an alkyl group containing from 1 to 3 carbon atoms. Medication with antagonist action on H2 receptors of histamine and antiulcer action, containing a thieno- or furo[2,3-c]pyrrole as active principle.</p>
申请公布号 IN169684(B) 申请公布日期 1991.12.07
申请号 IN1985DE88119 申请日期 1985.10.22
申请人 LIPHA LYONNAISE INDUSTRIELLE PHARMACEUTIQUE 发明人 FESTAL DIDIER;DESCOURS DESNIS;DEPIN JEAN-CLAUDE;QUENTIN YVETTE
分类号 A61K31/40;A61K31/4365;A61P1/04;C07D491/04;C07D491/048;C07D495/04;(IPC1-7):C07D209/60 主分类号 A61K31/40
代理机构 代理人
主权项
地址