发明名称 |
Synthesis of 4-amino-1,2-hydrocarbyl pyrazolidines via 4-nitro analogs |
摘要 |
4-Nitro-1,2-hydrocarbyl pyrazolidines are prepared by a novel route from 1,2-disubstituted hydrazines and 1,3-di-(secondary amino)-2-nitropropanes and reduced to the corresponding 4-amino-1,2-hydrocarbyl pyrazolidines, which latter compounds are intermediates in the preparation of certain pharmaceutical benzamides. The novel 4-nitro-1,2-hydrocarbyl pyrazolidines have the formula: <IMAGE> wherein R1 and R2 are selected from loweralkyl, lowercycloalkyl or phenyl-loweralkyl and may be the same or different.
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申请公布号 |
US4358599(A) |
申请公布日期 |
1982.11.09 |
申请号 |
US19810272806 |
申请日期 |
1981.06.11 |
申请人 |
A. H. ROBINS COMPANY, INC. |
发明人 |
LO, YOUNG S.;MUNSON, JR., HARRY R. |
分类号 |
C07D231/04;(IPC1-7):C07D231/04 |
主分类号 |
C07D231/04 |
代理机构 |
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