发明名称 FOERFARANDE FOER FRAMSTAELLNING AV NYA TERAPEUTISKT ANVAENDBARA N-(1-(ACYLOXIMETYL)-4-(OMEGA-NITROGUANIDINO)-BUTYL)-DIHYDROLYSERGAMIDER SAMT SYRAADDITIONSSALTER DAERAV
摘要 New compounds of the general formula (I) <IMAGE> (I) wherein R stands for hydrogen or methyl group, X Y STANDS FOR A GROUP OF THE FORMULA <IMAGE> and R1 stands for a group of the formula (III), (IV) or (V) <IMAGE> (III) <IMAGE> (IV) <IMAGE> (V) wherein n is an integer from 4 to 10, ARE PREPARED BY ACYLATING A COMPOUND OF THE GENERAL FORMULA (II), <IMAGE> (II) wherein R and x y each have the same meanings as defined above, and R2 stands for a group of the formula (VI), (VII) or (VIII), <IMAGE> (VI) <IMAGE> (VII) <IMAGE> (VIII) with a C6-12 carboxylic acid or a C6-12 carboxylic acid halide.
申请公布号 FI61897(C) 申请公布日期 1982.10.11
申请号 FI19750001537 申请日期 1975.05.27
申请人 RICHTER GEDEON VEGYESZETI GYAR R T 发明人 MAGO ERZSEBET;BORSI JOZSEF;CSANYI ENDRE;PIK KATALIN;WOLF LAJOS
分类号 A61K31/48;A61P25/24;A61P25/26;A61P43/00;C07D457/02;C07D457/06;(IPC1-7):C07D457/06 主分类号 A61K31/48
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