发明名称 NEW PROCESS FOR PREPARING IMIDAZOBENZODIAZERINES AND SALTS
摘要 Compounds of the general formula (I), <IMAGE> (in which R1 represents a hydrogen atom, a halogen atom, a nitro radical or a trifluoromethyl radical, R2 represents a hydrogen atom or a halogen atom and R3 and R4, together with the nitrogen atom to which they are attached, represent a 4-alkyl- piperazin-1-yl, 4-cycloalkyl-alkyl- piperazin-1-yl, 4-phenyl-piperazin-1-yl or piperidino radical) as well as their addition salts with mineral or organic acids, are prepared by reacting a compound of formula (II), <IMAGE> with an amine of formula III, <IMAGE> (in which alk and alk' represent alkyl radicals containing from 1 to 3 carbon atoms) in the presence of an organic solvent followed, if desired by salt formation.
申请公布号 AU8094782(A) 申请公布日期 1982.09.30
申请号 AU19820080947 申请日期 1982.02.26
申请人 ROUSSEL-UCLAF 发明人 JACQUES PROST-MARECHAL
分类号 C07D487/04 主分类号 C07D487/04
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