PROCESS FOR THE PREPARATION OF 3-(2-HYDROXY-4-(SUBSTITUTED)PHENYL)CYCLOALKANOL ANALGESIC AGENTS AND THEIR DERIVATIVES

摘要

Cycloalkanones, cycloalkanols and unsaturated analogs thereof, each of which has at the 3-position a 2-hydroxy-4-substituted phenyl group wherein the 4-position substituent is OH, alkyl which can have an oxygen atom as part of the chain, or aralkyl which can have an oxygen atom as part of the alkyl chain, are useful as CNS agents especially as analgesics, tranquilisers, sedatives and antianxiety agents and/or as anticonvulsants, diuretics and antidiarrheal agents.