发明名称 PHENYLCLOHEXANE DERIVATIVE
摘要 NEW MATERIAL:A phenylcyclohexane derivative of formula I(R<1> is H, hydroxyl group or alkoxyl; R<2> is H, aminoalkyl, alkoxylcarbonylalkyl or aminocarbonylalkyl; R<3> is oxo, hydroxyl group, alkylcarbonylamino, alkycarbonyloxy, aminoalkylcarbonyloxy, etc.; R<4> is H, aminoalkyl, morpholino or morpholinoalkyl; however, R<3> and R<4> are not H at the same time). EXAMPLE:2-Ethoxycarbonylmethyl-6-morpholino-2-phenylcyclohexanone. USE:Useful as a medicine having inhibitory action on blood platelet aggregation, inhibitory action on contraction of extirpated intestines and anti-inflammatory and analgesic actions. PROCESS:Either one of R<2> or R<4> or both are introduced into a phenylcyclohexane of formula II as a starting raw material by the well-known method to give the aimed compound of formulaI (R<3> is oxo group).
申请公布号 JPS57122041(A) 申请公布日期 1982.07.29
申请号 JP19810008493 申请日期 1981.01.21
申请人 SUNTORY KK 发明人 FUJIMURA HAJIME;HORI MIKIO;TATSUOKA TOSHIO;OKITSU MITSUTO;IMAO KAYOKO;MORITA MINORU
分类号 C07D295/08;A61K31/135;A61K31/16;A61K31/165;A61K31/215;A61K31/27;A61K31/445;A61K31/535;A61K31/5375;A61P7/02;A61P25/04;A61P29/00;C07C67/00;C07C69/03;C07C69/73;C07C213/00;C07C215/42;C07C215/64;C07C217/12;C07C217/74;C07C219/24;C07C225/18;C07C227/00;C07C229/08;C07C229/12;C07C229/34;C07C233/11;C07C233/23;C07C233/32;C07C233/38;C07C233/41;C07C235/34;C07C235/40;C07C235/78;C07C235/82;C07C237/20;C07C237/22;C07C237/24;C07D295/04;C07D295/12;C07D295/14 主分类号 C07D295/08
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