发明名称 |
DIURETIC COMPOSITIONS COMPRISING 2,4-DIAMINO-5-(4-AMINO-3,5-DIMETHOXYBENZYL)-PYRIMIDINE AND A DIURETIC WHICH CAUSES EXCRETION OF POTASSIUM AND THEIR PREPARATION |
摘要 |
<p>A composition having diuretic activity which contains a potassium-flushing diuretic and a potassium-retaining compound, said potassium-retaining compound is a compound of the formula <IMAGE> I wherein R1 and R2 are C1-6-alkyl or C2-6-alkenyl, and R3 and R4, independently, are hydrogen, C1-6-alkyl, C2-6-alkenyl or C1-6-acyl, or R3 and R4 together with the nitrogen atom are an optionally unsaturated 5-, 6- or 7-membered heterocyclic group, or a physiologically compatible salt thereof, are described.</p> |
申请公布号 |
EP0009657(B1) |
申请公布日期 |
1982.06.23 |
申请号 |
EP19790103328 |
申请日期 |
1979.09.07 |
申请人 |
F. HOFFMANN-LA ROCHE & CO. AKTIENGESELLSCHAFT |
发明人 |
DAUM, ADAM, DR.;FERNEX, MICHEL, DR.;WICK, ALEXANDER EDUARD, DR. |
分类号 |
C07D239/49;A61K31/505;A61K31/54;A61K31/55;A61P7/10;C07D403/10;(IPC1-7):61K31/54 |
主分类号 |
C07D239/49 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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