发明名称 UN PROCEDIMIENTO PARA LA PREPARACION DE CICLOALCA (4,5) PI- RROLO (2,3-G)-ISOQUINOLINAS
摘要 <p>The title compd. (I; R1 = alkyl, hydroxyalkyl, arylhydroxyalkyl, alkoxyalkyl, acyloxyalkyl, acylalkyl, aralkl, alkenyl, cycloalkyl- alkyl, alkynyl, thienyl-alkyl, furyl-alkyl, arylcarboxamidoalkyl, aralkenyl, alkenyloxyalkyl, aryloxyalkyl, aralkoxyalkyl, or aryl-N- imidazolonylalkyl; X = O or S; n = 3,4,5 or 6!, useful as a nervous sedative, was prepd. by the substitution of II in the presence of an isoquinoline N atom.</p>
申请公布号 ES499861(D0) 申请公布日期 1982.05.01
申请号 ES19610004998 申请日期 1981.02.27
申请人 F.HOFFMANN-LA ROCHE & CIE. S.A. 发明人
分类号 C07D471/04;A61K31/40;A61K31/47;A61P25/18;C07D;(IPC1-7):07D471/04;61K31/40;61K31/47 主分类号 C07D471/04
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