发明名称 Verfahren zur Herstellung von neuen Benzodiazepinen
摘要 1,179,125. Benzophenone derivatives. SCHERICO Ltd. 13 Jan., 1967 [14 Jan., 1966], No. 46993/69. Divided out of 1,179,124. Heading C2C. Compounds of the general formula (X=H, halogen, CF 3 , NO 2 , alkyl or alkoxy; Z=H or -COCR<SP>1</SP>R<SP>2</SP>L in which R<SP>1</SP>'<SP>2</SP>= H or alkyl and L=halogen or free or protected amino group; U = -COPh in which Ph = phenyl optionally substituted by halogen, CF 3 , NO 2 , alkyl or alkoxy) are prepared by standard methods, such as trifluoroethylation, acylation and the Friedel-Crafts reaction. The preparation of 2,2,2-trifluoroethyl trichloromethylsulphonate and of substituted N- (2,2,2-trifluoroethyl) anilines is described.
申请公布号 DE1695841(A1) 申请公布日期 1972.02.03
申请号 DE1967SC40084 申请日期 1967.01.13
申请人 SCHERICO LTD. 发明人 G. TOPLISS,JOHN
分类号 C07D243/16;C07D243/18;C07D243/24;C07D243/26;C07D243/28;C08G59/24 主分类号 C07D243/16
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