| 摘要 |
Phenyl-quinolizidines of the general formula <IMAGE> I wherein X is hydrogen, fluorine, chlorine, lower-alkoxy, lower-alkyl or trifluoromethyl; Y is hydrogen, fluorine, chlorine, lower-alkoxy or lower-alkyl; and R1 is acyl, acylamino or a group A of the formula <IMAGE> wherein R2 is oxygen or sulfur; R3 is hydrogen or lower-alkyl; and one of R4 and R5 is hydrogen and the other is bromine, iodine, cyano, lower-alkoxycarbonyl or sulfamoyl, as racemates or enatiomers, as well as acid addition salts thereof, utilizing various intermediates, are described. The foregoing compounds are useful as neuroleptic, antiemetic and analgesic agents. |
