发明名称 |
Process for the preparation of thiazine derivatives |
摘要 |
Thienothiazine derivatives of formula <IMAGE> wherein R2 denotes the radical of an aromatic heterocycle which has 1 to 4 heteroatoms and is optionally substituted by one or two lower alkyl groups or R2 denotes a phenyl radical which is optionally substituted in a particular manner defined in Claim 1, and R1, R3 and R4 have the meaning given in Claim 1, and salts thereof, have an anti-inflammatory, analgesic, antirheumatic and antithrombotic action. They may therefore be used as medicaments. The compounds of formula I are prepared by reacting corresponding compounds of formula <IMAGE> wherein R denotes lower alkyl, with appropriate amines of formula H2N-R2 IIIv
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申请公布号 |
CH624960(A5) |
申请公布日期 |
1981.08.31 |
申请号 |
CH19770000083 |
申请日期 |
1977.01.05 |
申请人 |
HOFFMANN-LA ROCHE, F., & CO. AG |
发明人 |
PROF. DR. DIETER BINDER;PROF. DR. OTTO HROMATKA;DR. RUDOLF PFISTER;DR. PAUL ZELLER |
分类号 |
C07D333/34;C07D333/38;C07D513/04;(IPC1-7):C07D513/04 |
主分类号 |
C07D333/34 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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