发明名称 |
PROCESS FOR PREPARING HETEROCYCLIC DERIVATIVES |
摘要 |
A process for manufacturing heterocyclic derivatives (I) used for effective antihistamines and antacids is described. Guanidine derivatives (1; X = S or NH: Y = O or S; m = 0-4: n = 1-4; R1 = H, halogen or C1-6 alkyl; R2 = H, C1-10 alkyl or C1-6 alkaloyl; A = 3,4-dioxocyclobutene-1,2-diol; B = C1-6 alkoxy) are prepared by reacting compound(II) and B-H compound.
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申请公布号 |
KR810000599(B1) |
申请公布日期 |
1981.06.05 |
申请号 |
KR19780001163 |
申请日期 |
1978.04.20 |
申请人 |
IMPERIAL CHEMICAL IND LTD;I C I AMERICAS INC |
发明人 |
GILMAN D;YELLIN T;JONES D;WARDLEWORTH J |
分类号 |
A61K31/415;A61K31/54;C07D233/88;C07D277/42;(IPC1-7):C07D277/42;A61K31/41 |
主分类号 |
A61K31/415 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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