发明名称 PROCESS FOR PREPARING THIAZOLIDINE CARBOXYLIC ACIDS AND RELATED ACIDES AND SALTS THEREOF
摘要 Title compds. (I; R = hydroxy or lower alkoxy; R1,R2 = H or lower alkyl; R5,R6 = H or lower alkyl; R3 = H, lower alkyl or mercapto-lower alkylene; R4 = H, lower alkanol, benzoyl or III; X = O, S, SO, or SO2; m = 1-3; n = 0-2; m+n = 2 or 3; P = O or 1) useful as inhibitors, were manufd. by acylation of II with R4S(CH2)pCHR3COOH.
申请公布号 KR810000464(B1) 申请公布日期 1981.05.09
申请号 KR19780001995 申请日期 1978.06.29
申请人 E R SQUIBB & SONS INC 发明人 ONDETTI M
分类号 A61K31/39;A61K31/42;C07D263/06;C07D277/06;C07D277/30;(IPC1-7):C07D263/06 主分类号 A61K31/39
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