发明名称 |
SUBSTITUIERTE TETRAAZATRICYCLEN, VERFAHREN ZU IHRER HERSTELLUNG, IHRE VERWENDUNG UND SIE ENTHALTENDE ARZNEIMITTEL |
摘要 |
1-(Lower)alkyl-4-(substituted)aminoalkylcarbonyl-1,4,9,10-tetrahydropy razolo[4,3-b][1,5]benzodiazepin-10-ones are useful, e.g., to protect warm blooded animals against the formation of gastric ulcers. They are active ingredients in otherwise conventional medicament compositions administered enterally or parenterally in standard dosage forms. Their synthesis, their novel intermediates and their acid-addition salts are described. |
申请公布号 |
DE3029281(A1) |
申请公布日期 |
1981.02.19 |
申请号 |
DE19803029281 |
申请日期 |
1980.08.01 |
申请人 |
BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH, 7750 KONSTANZ |
发明人 |
RAINER, GEORG, DIPL.-CHEM. DR.;RIEDEL, RICHARD, DR.;KLEMM, KURT, DIPL.-CHEM. DR., 7753 ALLENSBACH;ELTZE, MANFRID, DIPL.-CHEM. DR., 7750 KONSTANZ |
分类号 |
C07D487/04;A61K;A61K31/55;A61P1/04;C07D;C07D231/14;C07D231/16;C07D231/38 |
主分类号 |
C07D487/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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