发明名称 SUBSTITUTED ACETOPHENONES AND PROCESS THEREFOR
摘要 Antivirally active compounds of the formula <IMAGE> I wherein R1 represents hydroxy, acyloxy derived from an aliphatic acid having 2-18 carbon atoms or a heterocyclic carboxylic acid containing nitrogen atom(s), lower alkoxycarbonyloxy, aminoacyloxy or carboxyalkanoyloxy; R2 represents lower alkoxy; R3 represents hydrogen or lower alkoxy; and R4 represents phenyl which may be substituted by one or more substituents selected from the group consisting of lower alkyl, lower alkoxy, benzyloxy, allyloxy, alkylthio, dialkylamino, amino, cyano, hydroxy, halo and alkylenedioxy; or pyridyl, furyl, thienyl or pyrrolyl which may be substituted by lower alkyl, pharmaceutical compositions containing them and a process for the preparation of those compounds of formula I which are novel.
申请公布号 ZA8000312(B) 申请公布日期 1981.01.28
申请号 ZA19800000312 申请日期 1980.01.18
申请人 HOFFMANN LA ROCHE 发明人 MORIO FUJIU;HIDEO ISHITSUKA;YASUJI SUHARA
分类号 C07C69/035;A61K31/12;A61K31/135;A61K31/215;A61K31/22;A61K31/265;A61K31/27;A61K31/34;A61K31/341;A61K31/357;A61K31/36;A61K31/38;A61K31/40;A61K31/44;A61K31/4406;A61K31/4418;A61K31/455;A61P31/12;C07C45/00;C07C45/74;C07C49/84;C07C67/00;C07C69/353;C07C225/16;C07C239/00;C07C253/00;C07C255/47;C07C255/56;C07C271/06;C07C313/00;C07C319/20;C07C323/22;C07D207/32;C07D207/333;C07D213/50;C07D213/80;C07D241/24;C07D307/46;C07D317/54;C07D317/64;C07D333/22 主分类号 C07C69/035
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