发明名称 |
PROCESS FOR THE PRODUCTION OF ARYL UREAS |
摘要 |
<p>Urea derivatives of the formula (wherein Ar represents a residue of 5- or 6-membered heteroaromatic ring; R represents a hydrogen atom or a C1-C6 alkyl group; R1 represents a C1-C6 alkyl group; and R2 represents a C1-C6 alkyl, C2-C6 alkenyl, or C1-C6 alkoxy group) are produced by reacting an amine of the formula Ar-NH-R (wherein Ar and R have the significance given above) with a carbamoyl halogenide of the formula (wherein X represents a halogen atom, and R1 and R2 have the significance given above) in the presence of a Lewis acid in an inert solvent.</p> |
申请公布号 |
CA1093081(A) |
申请公布日期 |
1981.01.06 |
申请号 |
CA19780300467 |
申请日期 |
1978.04.05 |
申请人 |
SHIONOGI & CO. LTD. |
发明人 |
MAKISUMI, YASUO;SASATANI, TAKASHI;MURABAYASHI, AKIRA |
分类号 |
C07D275/02;C07D213/75;C07D261/14;C07D263/48;C07D275/03;C07D277/20;C07D277/38;C07D277/46;C07D277/48;C07D277/82;(IPC1-7):07D213/75;07D261/14;07D277/00 |
主分类号 |
C07D275/02 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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