发明名称 |
ИНГАЛЯЦИОННАЯ КОМПОЗИЦИЯ, СОДЕРЖАЩАЯ СУЛЬФОАЛКИЛОВЫЙ ЭФИР ЦИКЛОДЕКСТРИНА И КОРТИКОСТЕРОИД |
摘要 |
An inhalable unit dose liquid formulation containing SAE-CD and corticosteroid is provided. The formulation is adapted for administration to a subject by nebulization with any known nebulizer. The formulation can be included in a kit. The formulation is administered as an aqueóus solution or concentrated composition. The formulation is employed in an improved nebulization system for administering corticosteroid by inhalation. SAE-CD present in the formulation significantly enhances the chemical stability of corticosteroid, such as budesonide. A method of administering the formulation by inhalation is provided. The formulation can also be administered by conventional nasal delivery apparatus. The formulation is prepared by mixing SAE-CD, in solid or liquid (dissolved) form, with an inhalable suspension-based unit dose formulation. |
申请公布号 |
RU2006127443(A) |
申请公布日期 |
2008.02.10 |
申请号 |
RU20060127443 |
申请日期 |
2004.12.31 |
申请人 |
САЙДЕКС, ИНК. (US) |
发明人 |
ПИПКИН Джеймс Д. (US);ЦИММЕРЕР Руперт О. (US);ТОМПСОН Дайан О. (US);МОШЕР Джерольд Л. (US) |
分类号 |
A61K9/12;A61K9/00;A61K9/08;A61K9/14;A61K31/16;A61K31/57;A61K31/715;A61K47/40;A61K47/48;C08B37/16 |
主分类号 |
A61K9/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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