发明名称 Phthalazine cardiac stimulants, processes for preparing them, and pharmaceutical compositions containing them.
摘要 <p>Phthalazine cardiac stimulants of the formula &lt;CHEM&gt; wherein R&lt;1&gt; is a C1-C4 alkyl group, and Y is a group of the formula: -(CH2)m-Z, wherein m is 1 or 2, and Z is a group selected from: -OCONR&lt;3&gt;R&lt;4&gt;, -N(R&lt;2&gt;)COR&lt;3&gt;, -N(R&lt;2&gt;)SO2R&lt;3&gt;, -N(R&lt;2&gt;)CONR&lt;3&gt;R&lt;4&gt;, -N(R&lt;2&gt;)SO2NR&lt;3&gt;R&lt;4&gt;, and -N(R&lt;2&gt;)COOR&lt;3&gt;, wherein R&lt;2&gt; and R&lt;4&gt; are each independently hydrogen or C1-C4 alkyl, and R&lt;3&gt; is C3-C7 cycloalkyl; or a pharmaceutically acceptable acid addition salt thereof. Also described are processes for preparing the compounds and pharmaceutical compositions containing them.</p>
申请公布号 EP0017411(A1) 申请公布日期 1980.10.15
申请号 EP19800300909 申请日期 1980.03.24
申请人 PFIZER LIMITED;PFIZER CORPORATION 发明人 CAMPBELL, SIMON FRASER;DANILEWICZ, JOHN CHRISTOPHER;HAM, ALLAN LESLIE;STUBBS, JOHN KENDRICK
分类号 C07D213/42;C07D401/04;A61K31/50;A61P9/04;C07D211/22;C07D211/26;C07D211/28;C07D213/30;C07D213/40;(IPC1-7):07D401/04;61K31/495 主分类号 C07D213/42
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