发明名称 ACID ADDITION SALTS OF 16 BETA -MONOQUATERNARY AMMONIUM DERIVATIVES OF 2 BETA,16 BETA-BIS-PIPERIDINO-ANDROSTANES AND PHARMACEUTICAL PREPARATIONS CONTAINING SAME
摘要 New and pharmacologically useful pharmaceutically acceptable acid addition salts are disclosed for the 16 beta -mono-quaternary ammonium derivatives of either the 2 beta , 16 beta -bis-piperdino-3- alpha , 17 beta -dihydroxy-5 alpha -androstane 3 alpha , 17 beta -di-lower aliphatic esters of the 2 beta , 16 beta -bis-piperidino-3 alpha -hydroxy-5 alpha -androstane-3 alpha -lower aliphatic esters, which salts are surprisingly relatively stable in aqueous solutions, so that they provide stable aqueous injection preparations.
申请公布号 ZA7904371(B) 申请公布日期 1980.08.27
申请号 ZA19790004371 申请日期 1979.08.20
申请人 AKZO NV 发明人 SAVAGE D;CARLYLE I;SLEIGH T
分类号 A61K31/58;A61P25/02;C07J43/00 主分类号 A61K31/58
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