发明名称 |
PROCESS FOR THE PREPARATION OF AMINOGLYCOSIDE ANTIBIOTICS AND NOVEL INTERMEDIATES THEREFOR |
摘要 |
<p>A process for preparing 1-N-substituted kanamycin A or B derivatives which comprises acylation or alkylation of selectively N-protected intermediate compounds and a process for preparing the novel selectively N-protected intermediate compounds.</p> |
申请公布号 |
CA1083568(A) |
申请公布日期 |
1980.08.12 |
申请号 |
CA19770276055 |
申请日期 |
1977.04.13 |
申请人 |
PFIZER CORPORATION |
发明人 |
MILLION, WILLIAM A.;PLEWS, RHONA M.;RICHARDSON, KENNETH |
分类号 |
C07H15/234;A61K31/70;A61K31/7028;A61K31/7034;A61K31/7036;A61P31/04;C07H15/236;(IPC1-7):07H15/22 |
主分类号 |
C07H15/234 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|