| 摘要 |
1. Substituted N-propargyl-anilines of the general formula see diagramm : EP0010673,P37,F3 in which R**1 , R**2 , R**3 , R**4 and R**5 represent hydrogen and alkyl with 1 to 4 carbon atoms, and furthermore R**1 additionally represents halogen and R**5 additionally represents phenyl which is optionally substituted by halogen, alkyl with 1 to 4 carbon atoms and nitro, and halogen, R**6 represents tetrahydrofuryl, thiophenyl, tetrahydrothiophenyl, optionally methyl- or ethyl-substituted isoxazolyl, and optionally cyano- or thiocyano-substituted alkyl with 1 to 4 and alkenyl and alkinyl each with 2 to 4 carbon atoms, and represents the groupings -CH2 -Az, -CH2 -OR**8 , -CH2 -SR**7 , -OR**7 , -CH2 -OSO2 R**8 , -COOR**7 and see diagramm : EP0010673,P38,F1 wherein R**7 and R**8 represent halogen-, cyano and thiocyano-substituted alkyl with 1 to 4 carbon atoms and alkenyl and alkinyl, with in each case 2 to 4 carbon atoms, which are optionally substituted by the indicated alkyl substituents and represents alkoxyalkyl with 1 to 4 carbon atoms in each alkyl part, and furthermore R**7 can additionally represent unsubstituted alkyl with 1 to 4 carbon atoms, and Az represents pyrazol-1-yl) 1,2,4-triazol-1-yl and imidazol-1-yl. |
