发明名称 |
Derivatives of 2-oxazolydone and methods for preparing the same |
摘要 |
A compound having pharmacological properties comprising the structural formula <IMAGE> (I) wherein R is selected from the isopropyl, n-octyl, n-butyl or isobutyl groups; R1 is selected from the 1-naphthyloxymethyl, (2-allylphenoxy)-methyl, 4-nitrophenyl, {2-[(tetrahydrofurfuryl)oxy-]-phenoxy}-methyl, [4-(2-methoxyethyl)phenoxy]methyl, 4-isopropylthiophenyl, 4-acetaminophenoxymethyl groups; and R2 represents a hydrogen atom or a methyl group. A method for synthetizing the compound is also disclosed comprising the cyclization of aminoalcohol or halogenurethane.
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申请公布号 |
US4188323(A) |
申请公布日期 |
1980.02.12 |
申请号 |
US19780905047 |
申请日期 |
1978.05.11 |
申请人 |
MENARINI A., S.A.S. |
发明人 |
BIANCHINI, CLAUDIO;GHELARDONI, MARIO;MELI, ALBERTO;PESTELLINI, VITTORIO;SOLDATO, PIERO DEL;VOLTERRA, GIOVANNA |
分类号 |
A61K31/42;A61K31/421;A61P9/08;A61P25/02;C07D263/20;C07D263/24;C07D413/12;(IPC1-7):C07D263/24 |
主分类号 |
A61K31/42 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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