| 摘要 |
The title cmpds. [I; X = C1-6 alkyl, C4-7 cycloalkyl, C2-5 hydroxyalkyl or C1-5 phenoxyalkyl; R = H, halogen, nitro, amino or methylthio; R1,R2 = H were prepd. by the reaction, of II and Hal-X[X = X' or X"; X' = tetrahydropyranyloxyalkyl; X" = C1-6 alkyl, C5-6 cycloalkylthio 3-(1,2,3,6-tetrahydro-4-pyridyl)-1Hindole HCl salt, 4.2cm3 propyliodide, 6g sodium carbonate and 160cm3 dimethylformamide was stirred for 4 hrs. and crystallized to give 5.2 g 5-methyltio-3-(1-propyl-1,2,3,6-tetrahydro-4-pyridyl)1H-indole HCl salt.
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