发明名称 HETEROCYKLISKE DERIVATER AF (4-PHENYLPIPERANZIN-1-YL-ARYLOXYMETHYL-1,3-DIOXOLAN-2-YL)-METHYL-1-H-IMIDAZOLER OG 1H-1,2,4-TRIAZOLER
摘要 1H-Imidazole and 1H-1,2,4-triazole derivatives of the formula <IMAGE> in which Q denotes CH or N, Ar denotes phenyl, thienyl, halogenthienyl or phenyl which is substituted by from 1 to 3 substituents selected from halogen, lower alkyl, lower alkoxy and trifluoromethyl, and Y is selected specifically from 1H-pyrrol-1-yl, 1H-pyrazol-1-yl, 1H- imidazol-1-yl, 1H-1,2,4-triazol-1-yl, 4H-1,2,4-triazol-4- yl, 2,3-dihydro-4H-1,2,4-triazol-4-yl and 1H-1,2,3,4- tetrazol-1-yl radicals, or acid addition salts and stereochemically isomeric forms thereof, are prepared by a number of different processes. The compounds possess antifungal and antibacterial activity. Compounds of the formula <IMAGE> can be used as intermediates for preparing compounds of the formula I and also possess antifungal and antibacterial activity. <IMAGE>
申请公布号 DK261479(A) 申请公布日期 1979.12.24
申请号 DK19790002614 申请日期 1979.06.21
申请人 JANSSEN PHARMACEUTICA N V 发明人 HEERES J;BACKX L J J
分类号 A01N;A01N43/50;A01N43/60;A01N43/64;A61K31/335;A61K31/41;A61K31/495;C07D;C07D207/32;C07D231/50;C07D233/00;C07D233/60;C07D239/00;C07D249/04;C07D249/08;C07D257/04;C07D295/12;C07D317/28;C07D405/12;C07D405/14;C07D409/14;(IPC1-7):C07D/ 主分类号 A01N
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