发明名称 THIOALKANOYLALKANOIC ACID COMPOUNDS
摘要 Thioalkanoylalkanoic acid compounds and salts thereof having the formula <IMAGE> wherein R1, R2, R3 and R4 each is hydrogen or lower alkyl; R5 is hydrogen, lower alkanoyl, benzoyl or <IMAGE> A and B each is hydrogen or join together as a polymethylene chain -(CH2)n- to complete a 4-, 5- or 6- membered cycloalkyl group, and m is 0 or 1, are angiotensin converting enzyme inhibitors and are useful as hypotensive agents.
申请公布号 AU4260478(A) 申请公布日期 1979.10.04
申请号 AU19780042604 申请日期 1978.12.15
申请人 SQUIBB, E.R. & SONS, INC. 发明人 MIGUEL ANGEL ONDETTI;MICHAEL EDWARD CONDON
分类号 A61K31/19;A61K;A61K31/10;A61K31/21;A61K31/215;A61K31/22;A61K31/265;A61P9/12;C07C;C07C59/76;C07C61/00;C07C61/08;C07C61/16;C07C67/00;C07C69/74;C07C313/00;C07C323/52;C07C323/53;C07C325/00;C07C327/20;C07C327/22;C07C327/32;C07D307/93 主分类号 A61K31/19
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