发明名称 |
THIOALKANOYLALKANOIC ACID COMPOUNDS |
摘要 |
Thioalkanoylalkanoic acid compounds and salts thereof having the formula <IMAGE> wherein R1, R2, R3 and R4 each is hydrogen or lower alkyl; R5 is hydrogen, lower alkanoyl, benzoyl or <IMAGE> A and B each is hydrogen or join together as a polymethylene chain -(CH2)n- to complete a 4-, 5- or 6- membered cycloalkyl group, and m is 0 or 1, are angiotensin converting enzyme inhibitors and are useful as hypotensive agents. |
申请公布号 |
AU4260478(A) |
申请公布日期 |
1979.10.04 |
申请号 |
AU19780042604 |
申请日期 |
1978.12.15 |
申请人 |
SQUIBB, E.R. & SONS, INC. |
发明人 |
MIGUEL ANGEL ONDETTI;MICHAEL EDWARD CONDON |
分类号 |
A61K31/19;A61K;A61K31/10;A61K31/21;A61K31/215;A61K31/22;A61K31/265;A61P9/12;C07C;C07C59/76;C07C61/00;C07C61/08;C07C61/16;C07C67/00;C07C69/74;C07C313/00;C07C323/52;C07C323/53;C07C325/00;C07C327/20;C07C327/22;C07C327/32;C07D307/93 |
主分类号 |
A61K31/19 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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