发明名称 2-Methoxy-benzamide derivatives
摘要 The invention provides novel 2-methoxy-benzamide derivatives of the formula: <IMAGE> (I) in which n is 1 or 2; R1 represents a cycloalkyl-alkyl radical of formula: <IMAGE> a phenylalkyl radical of formula <IMAGE> (in which m is an integer from 2 to 5, A is a linear or branched alkylene chain of 1 to 4 carbon atoms, and R4 is hydrogen, halogen, especially fluorine or chlorine, trifluoromethyl, or alkyl or alkoxy of 1 to 3 carbon atoms), CNCH2-CH2-, CH 3BOND C-CH2-, <IMAGE> R2 is either chlorine, SO2 R5 (in which R5 is alkyl of 1 to 4 carbon atoms), or SO2NR6R7 (in which, R6 and R7, which are identical or different, represent, independently of one another, hydrogen or alkyl of 1 to 4 carbon atoms); and R3 is hydrogen or alkyl of 1 to 4 carbon atoms; in the form of racemates or optical isomers, and their pharmaceutically acceptable acid addition salts, which are useful in the treatment of psychosomatic and psychotic disturbances.
申请公布号 US4158060(A) 申请公布日期 1979.06.12
申请号 US19760749282 申请日期 1976.12.10
申请人 SYNTHELABO S.A. 发明人 GIUDICELLI, DON P R L;JALFRE, MAURICE;KAPLAN, JEAN-PIERRE;MANOURY, PHILIPPE M J;NAJER, HENRY;OBITZ, DANIEL C L;RAIZON, BERNARD M
分类号 C07D207/08;C07D207/20;C07D207/26;C07D207/263;C07D207/27;C07D211/26;C07D211/70;C07D211/76;(IPC1-7):C07D207/08;A61K31/40 主分类号 C07D207/08
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