| 摘要 |
<p>(A) O-Indolylglycolic acids and derivs., (I) where A = an acyl group derived from an opt. substd. aromatic or heterocyclic carboxylic acid, pref. with less than 3 rings. R' = H or a (1-8 C) hydrocarbon residue, e.g. alkyl or aryl opt. substd. by alkoxy or halogen, or aralkyl. R2 = H, Ph or alkyl R3 = H, halogen, CF3, alkyl or alkoxy. R4 = H, halogen, OH, alkyl, haloalkyl, aryl, alkylO-, arylO-, aralkylO-, cycloalkyl O-, alkenyl O-, NH2, NH alkyl, N alkyl2, NH aryl, alkyl-arylamino, CN, NO2, SH, -S alkyl, or -S aralkyl. M = OH, opt. substd. NH2, alkyl O-, alkenyl O-, cyclicalkoxy, aryl O-(all opt. substd.), or OY, where Y is cation or is (B) Acid addn. salts of (I). Anti-inflammatories and anti-pyretics. Dose 1.0-2,000 mg./day.</p> |
