发明名称 EBURNAMENINE DERIVATIVES
摘要 Derivatives of eburnamenine, of formula: <IMAGE> in which R1 = H and R2 = OH or R1 + R2 = additional bond; R3 = COOR4 (with R4 = alkyl containing 2 to 6 carbon atoms or a cycloalkyl) or CONR5R6. Or R1 = R2 = H and R3 = COOR7 (with R7 = alkyl containing 1 to 6 carbon atoms or a cycloalkyl) or CONR5R6, R5 and R6 = H, alkyl, cycloalkyl or form a heterocyclic radical together with the nitrogen atom. The first stage of their preparation is a bromination. The compounds have an antianoxic and psychotropic activity.
申请公布号 AU4129978(A) 申请公布日期 1979.05.17
申请号 AU19780041299 申请日期 1978.11.02
申请人 SYNTHELABO 发明人 GABOR ISTVAN KOLETAR;HENRY NAJER;PATRICK ANDRE LOUIS LARDENOIS;JEAN PIERRE LEFEVRE
分类号 A61K31/435;A61P9/08;A61P25/26;C07D461/00 主分类号 A61K31/435
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