发明名称 |
FORFARANDE FOR FRAMSTELLNING AV MAYTANSINOIDER |
摘要 |
Maytansinoid compounds are produced by contacting in the presence of a carbodiimide the compound maytansinol <IMAGE> with an acid of the formula: <IMAGE> (II) wherein R is lower alkyl, to yield the desired maytansinoids HAVING THE RESULTANT FORMULA: <IMAGE> (I) wherein R is lower alkyl. |
申请公布号 |
SE7811689(A) |
申请公布日期 |
1979.05.15 |
申请号 |
SE19780011689 |
申请日期 |
1978.11.13 |
申请人 |
* TAKEDA CHEMICAL INDUSTRIES LTD |
发明人 |
N * HASHIMOTO;T * KISHI |
分类号 |
C07D498/04;C07D498/18;(IPC1-7):C07D498/08 |
主分类号 |
C07D498/04 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|