发明名称 PROCEDIMENTO PER PREPARARE ACIDO (S-5S)-AMMINO-3-CLOROISOSSAZOLINA-5ACETICO E SUOI ANALOGHI E PRODOTTO OTTENUTO
摘要 <p>Analogues of AT-125 having the formula <IMAGE> wherein R is hydrogen, alkyl, haloalkyl or aralkyl; X is halogen, alkoxy, alkylthio, aryloxy, arylthio, aralkoxy, aralkythio, amino, alkylamino or dialkylamino; and NR14R15 is amino or a blocked amino group, provided that X is not chlorine when R is hydrogen or alkyl and R14 or R15 is alkoxycarbonyl or NR14R15 is phthalimido. The analogues can have therapeutic activity. AT-125 and the analogues can be prepared by halogenation of a corresponding analogue of tricholomic acid.</p>
申请公布号 IT7949040(D0) 申请公布日期 1979.05.14
申请号 IT19790049040 申请日期 1979.05.14
申请人 THE UPJOHN COMPANY SOCIETA' DELLO STATO DEL DELAWARE 发明人
分类号 A61K31/42;A61P31/04;C07D209/48;C07D261/04;C07D261/10;C07D261/12;C07D261/14;C07D303/04;C07D413/04;C07D413/06;(IPC1-7):A61K/ 主分类号 A61K31/42
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