发明名称 N'-(AMINOACYLAMINOPHENYL) ACETAMIDINES AND A METHOD FOR THEIR PREPARATION
摘要 <p>A new class of N'-(aminoacylaminophenyl) acetamidines: in which R1 and R2 are the same or different and represent hydrogen, alkyl, aryl or the substituted derivatives thereof or, together with the nitrogen atom to which they are attached, an heterocyclic ring; and R3 is hydrogen, alkyl, aryl, aralkyl, or a heterocyclic moiety including the substituted derivatives thereof. The products have utility as anthelmintics. The products are obtained by treating a suitable amino-acid or a carbonyl-activated amino-acid, with the appropriate N'-(4-aminophenyl)-N,N-dimethylacetamidine. In addition, the products are obtained by treating a suitable N'-(haloacylaminophenylacetamidine with an appropriate amine.</p>
申请公布号 CA1050022(A) 申请公布日期 1979.03.06
申请号 CA19740209256 申请日期 1974.09.16
申请人 BAYER AKTIENGESELLSCHAFT 发明人 WOLLWEBER, HARTMUND;NIEMERS, EKKEHARD;SCHULZ, HANS P.;THOMAS, HERBERT;ANDREWS, PETER
分类号 A61K31/165;A61K31/155;A61K31/40;A61K31/495;A61K31/535;C07C67/00;C07C231/00;C07C231/02;C07C231/12;C07C239/00;C07C257/14;C07C257/20;C07D295/15;(IPC1-7):07C123/00;07D295/14 主分类号 A61K31/165
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