FORFARANDE ATT MEDELST EN DIELS-ALDER-KONDENSATION FRAMSTELLA TRICYKLISKA DIKARBOXIMIDER MED VERDEFULLA TERAPEUTISKA EGENSKAPER

摘要

Tricyclicdicarboximides representatively prepared by the Diels-Alder condensation of a cyclic diene such as cycloheptatriene, cyclooctatetraene and the like with a dienophile such as substituted N-phenylmaleimide and the like are disclosed having pharmaceutical utility as minor tranquilizers and anti-convulsants. Also disclosed are processes for the preparation of such tricyclicdicarboximides; pharmaceutical compositions comprising such compounds and their salt, ester and amide derivatives; and methods of treatment comprising administering such compounds and compositions.