发明名称 |
HETEROCYCLIC BIPHENYLYLAMIDES USEFUL AS 5HT1D ANTAGONISTS |
摘要 |
A compound of formula (I) or a salt thereof, wherein P is a 5 to 7-membered heterocyclic ring containing 1 to 3 heteroatoms selected from oxygen, nitrogen or sulphur; A is CONH or NHCO; B is oxygen, S(O)p where p is O, 1 or 2, or NR12; m is 1 to 4; and the R's are hydrogen or substituents, is useful as a 5HT1D receptor antagonist in the treatment of CNS disorders.
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申请公布号 |
WO9515954(A1) |
申请公布日期 |
1995.06.15 |
申请号 |
WO1994EP03948 |
申请日期 |
1994.11.28 |
申请人 |
SMITHKLINE BEECHAM PLC;GASTER, LARAMIE, MARY;KING, FRANCIS, DAVID;WYMAN, PAUL, ADRIAN |
发明人 |
GASTER, LARAMIE, MARY;KING, FRANCIS, DAVID;WYMAN, PAUL, ADRIAN |
分类号 |
A61K31/34;A61K31/341;A61K31/40;A61K31/41;A61K31/42;A61K31/4245;A61K31/425;A61K31/426;A61K31/44;A61K31/4402;A61K31/4406;A61K31/4418;A61K31/445;A61K31/495;A61K31/496;A61K31/505;A61K31/535;A61K31/5377;A61P5/00;A61P9/12;A61P13/02;A61P15/00;A61P25/00;A61P25/18;A61P25/24;A61P25/26;A61P25/28;C07D213/56;C07D239/26;C07D241/12;C07D249/08;C07D257/04;C07D261/08;C07D271/06;C07D271/10;C07D271/107;C07D277/28;C07D277/30;C07D307/38;C07D413/12;C07D521/00;(IPC1-7):C07D271/06;C07D271/07 |
主分类号 |
A61K31/34 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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