发明名称 PROCEDIMIENTO PARA LA PREPARACION DE NUEVOS 2,5-DIHIDRO-1,2-TIAZINO (5,6-B)INDOL-3-CARBOXAMIDO-1,1-DIOXIDOS.
摘要 <p>Compounds of the formula <IMAGE> WHEREIN R1 is hydrogen, methyl or ethyl; R2 is methyl or ethyl; Y is hydrogen, fluorine, chlorine, bromine, methoxy, methyl, ethyl or trifluoromethyl; and Ar is 2-thiazolyl which may have one or two methyl or ethyl substituents attached thereto; 5,6-dihydro-4H-cyclopentathiazol-2-yl; 4,5,6,7-tetrahydro-2-benzothiazolyl; 2-benzothiazolyl; 3-isothiazolyl which may have a methyl substituent attached thereto; 2-pyridyl which may have a methyl or hydroxyl substituent attached thereto; 3-pyridyl; 4-pyridyl; 4-pyrimidinyl; pyrazinyl; 2-benzimidazolyl; 2-oxazolyl which may have a methyl substituent attached thereto; 2-benzoxazolyl; or phenyl which may have a fluoro, chloro, bromo, methyl, ethyl, trifluoromethyl or methoxy substituent attached thereto; and non-toxic, pharmacologically acceptable salts thereof formed with inorganic or organic bases. The compounds as well as their salts are useful as antiphlogistics and blood platelet aggregation inhibitors.</p>
申请公布号 ES469112(A1) 申请公布日期 1978.11.16
申请号 ES19120004691 申请日期 1978.04.25
申请人 DR. KARL THOMAE GESELLSCHAFT MIT BES. HAFTUNG 发明人
分类号 A61K31/54;A61P7/02;A61P29/00;C07D209/42;C07D513/04;C07D513/14;(IPC1-7):07D/;61K/ 主分类号 A61K31/54
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