发明名称 NEW 3-AMINO-17A-AZA-D-HOMOANDROSTANE DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
摘要 The invention relates to new 3-amino-17a-aza-D-homo-5 alpha -androstane derivatives of the general formula I <IMAGE> I wherein R1 represents a methylene or an >N-CH3 group, and n stands for 1 or 2, and the acid addition salts and the quaternary salts of the general formula <IMAGE> I(a) thereof, wherein R2 stands for an alkyl or alkenyl group having from 1 to 4 carbon atoms, and A represents a halogen atom, provided that if R1 stands for an >N-CH3 group, R2 is attached to the nitrogen of that >N-CH3 group. The new compound possess a non-polarizing neuromuscular blocking activity and have a short activity period.
申请公布号 IL55352(D0) 申请公布日期 1978.10.31
申请号 IL19780055352 申请日期 1978.08.14
申请人 RICHTER GEDEON VEGYESZET 发明人
分类号 C07D221/18;A61K31/395;A61P21/02;C07J73/00 主分类号 C07D221/18
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