发明名称 |
FORENING FOR FRAMSTELLNING AV CEFALOSPORANSYRADERIVAT |
摘要 |
1473672 Cephalosporin derivatives FUJISAWA PHARMACEUTICAL CO Ltd 9 May 1974 [10 May 1973 6 July 1973 3 Dec 1973 10 Jan 1974 7 Feb 1974 8 Feb 1974 27 March 1974] 20637/74 Heading C2C Novel compounds I (in which R 1 is NO 2 , alkoxy, alkylsulphonamido, or alkylaminosulphonamido; R 2 is H or OH and must be OH if R 1 is NO 2 or alkoxy; R 3 is H or optionally alkylated heterocyclylthio provided R 3 is H if R 1 is alkoxy and R 2 is OH; X is amino or protected amino and M is H or a non-toxic cation) and their derivatives at the carboxyl group are prepared by reaction of a compound II with a compound III or by reaction of a compound IV in which R 3 <SP>11</SP> is alkanoyl and R 1 <SP>1</SP> is as R 1 except that it may not be alkoxy, with a thiol R 3 <SP>1</SP>H in which R 3 <SP>1</SP> is heterocyclylthio. Pharmaceutical compositions having antibacterial properties comprise a compound I together with a suitable carrier or diluent. |
申请公布号 |
SE7810360(A) |
申请公布日期 |
1978.10.03 |
申请号 |
SE19780010360 |
申请日期 |
1978.10.03 |
申请人 |
* FUJISAWA PHARAMACEUTICAL CO LTD |
发明人 |
T * KAMIYA;K * TANAKA;Y * SAITO;T * KISHIMOTO;H * YAZAWA;T * TERAJI;K * TAKAI;Y * NAKAI |
分类号 |
C07D501/06;A61K31/545;A61K31/546;C07C275/42;C07C335/22;C07D501/20;C07D501/22;C07D501/36;(IPC1-7):C07C143/72 |
主分类号 |
C07D501/06 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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