发明名称 FLUOROPYRIMIDINE DEIVATIVES
摘要 PURPOSE:Fluoropyrimidine derivatives of formula I(X is O, NH;R1 is OH or SH, etherified or not etherified, amino which may be substituted;R2 and R3 are H, lower alkyl, 2-tetrahydrofuryl, Y is esterified or amidated carboxyl, CN), e.g. methyl-5-fluoro-6-hydroxy-1,2,3,4,5,6-hexahydro-2,4-dioxopyrimidine-5c arboxylate.
申请公布号 JPS5353672(A) 申请公布日期 1978.05.16
申请号 JP19760129932 申请日期 1976.10.27
申请人 TAKEDA CHEMICAL INDUSTRIES LTD 发明人 MIYASHITA OSAMU;MATSUMURA KOUICHI;SHIMAZU HIROSHI;HASHIMOTO NAOTO
分类号 C07D239/22;A61K31/505;A61K31/513;A61P31/12;A61P35/00;C07D239/54;C07D405/04 主分类号 C07D239/22
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