发明名称 AMINO ACID DERIVATIVE
摘要 <p>Amino-acid derivatives of the formula I R1-CpH2p-(NH)q-CO-NH-CHR<2>-CO-Z-CmH2m-CHWR<3>-CO-NH-CHR<SP >3-CR<4>-(CHR<5>)n- CO-E-Q-Y 1 in which R<1> to R<5>, p, q, Z, m, n, E, Q, W and Y have the meanings given in Claim 1, and the salts thereof inhibit the activity of human plasma renin.</p>
申请公布号 JPH03148248(A) 申请公布日期 1991.06.25
申请号 JP19900250420 申请日期 1990.09.21
申请人 MERCK PATENT GMBH 发明人 HORUSUTO JIYURASUJITSUKU;PEETAA RADATSUTSU;YOHANESU SONBUREEKU;YOAHIMU GANTE;KURAUSU YOTSUTO SHIYUMITSUCHIESU;KURAUSUUOTSUTOO MINKU
分类号 C07D295/04;A61K31/41;A61K31/44;A61K31/4402;A61K31/4406;A61K31/4409;A61K31/4412;A61K31/4418;A61K31/4427;A61K31/445;A61K31/4468;A61K31/495;A61K31/505;A61K38/00;A61P9/12;A61P43/00;C07C237/22;C07C271/22;C07C275/14;C07C275/16;C07C279/12;C07C281/06;C07C311/39;C07C323/59;C07C323/60;C07D211/36;C07D213/56;C07D233/54;C07D239/42;C07D241/20;C07D257/04;C07D257/06;C07D295/15;C07D401/12;C07K1/02;C07K1/113;C07K5/02;C07K5/06;C07K14/81 主分类号 C07D295/04
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