| 摘要 |
Title compds. (I; R = halogen, nitro, lower alkyl, lower alkoxy, hydroxy or H; R1 = H, lower alkyl, lower alkenly, or =CH2(CH2)pR2; R2 = arom. alkyl, cyclic lower alkyl; p = 0-3; n = 1-5) were prepd. by the reaction of II and III(X = halogen). Thus, 6.0 g (-)-3-hydroxy-N-methylmorphinan, 4.8 g potassium carbonate, 9.0 g hexafluorobenzene and 6.0 g Cu were reacted at 120≦̸C for 7 days in 60 ml pyridine to give I.
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