发明名称 SYNTHESIS OF INTERMEDIATES IN THE PREPARATION OF ACAT INHIBITORS.
摘要 <p>PCT No. PCT/US91/08758 Sec. 371 Date Sep. 13, 1993 Sec. 102(e) Date Sep. 13, 1993 PCT Filed Nov. 27, 1991 PCT Pub. No. WO92/13843 PCT Pub. Date Aug. 20, 1992.This invention relates to novel processes for synthesizing intermediates in the preparation of N-aryl and N-heteroarylamide inhibitors of the enzyme acyl coenzyme A: cholesterol acyltransferase (ACAT), and to novel intermediates used in such processes.</p>
申请公布号 GR3017357(T3) 申请公布日期 1995.12.31
申请号 GR19950402472T 申请日期 1995.09.13
申请人 PFIZER INC. 发明人 KELLY, SARAH, E.;CHANG, GEORGE
分类号 C07C69/14;A61K31/44;A61K31/47;C07C53/19;C07C59/01;C07C69/675;C07C211/27;C07C309/66;C07C309/73;C07C323/52;C07C323/60;C07D213/75;C07D215/00;C07D215/38;C07D217/02;C12P7/42;C12P7/62;C12P41/00;(IPC1-7):C07D215/38 主分类号 C07C69/14
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