发明名称 |
SYNTHESIS OF INTERMEDIATES IN THE PREPARATION OF ACAT INHIBITORS. |
摘要 |
<p>PCT No. PCT/US91/08758 Sec. 371 Date Sep. 13, 1993 Sec. 102(e) Date Sep. 13, 1993 PCT Filed Nov. 27, 1991 PCT Pub. No. WO92/13843 PCT Pub. Date Aug. 20, 1992.This invention relates to novel processes for synthesizing intermediates in the preparation of N-aryl and N-heteroarylamide inhibitors of the enzyme acyl coenzyme A: cholesterol acyltransferase (ACAT), and to novel intermediates used in such processes.</p> |
申请公布号 |
GR3017357(T3) |
申请公布日期 |
1995.12.31 |
申请号 |
GR19950402472T |
申请日期 |
1995.09.13 |
申请人 |
PFIZER INC. |
发明人 |
KELLY, SARAH, E.;CHANG, GEORGE |
分类号 |
C07C69/14;A61K31/44;A61K31/47;C07C53/19;C07C59/01;C07C69/675;C07C211/27;C07C309/66;C07C309/73;C07C323/52;C07C323/60;C07D213/75;C07D215/00;C07D215/38;C07D217/02;C12P7/42;C12P7/62;C12P41/00;(IPC1-7):C07D215/38 |
主分类号 |
C07C69/14 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|