Benzoxazinone amides as mineralocorticoid receptor modulators

摘要

Disclosed are certain derivatives of benzoxazinone amides of formula (I), or pharmaceutically acceptable salts thereof,;
that act as mineralocorticoid (MR) receptor modulators that may reduce oxidative stress in endothelium and hence improve vascular function, to methods for their potential therapeutic use, to pharmaceutical compositions containing them and to processes for preparing such compounds.

主权项

1. A compound of formula (I) wherein R1 is selected from CONH2 or CONHCH3; and R2 is selected from H, F, Cl or Br; or a pharmaceutically acceptable salt thereof.